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  • Pfizer's Xeljanz XR (once a day), approved in Korea
  • by | translator Choi HeeYoung | Dec 14, 2020 05:58am
JAK inhibitor Xeljanz XR, approved to treat rheumatoid arthritis
BID ¡æ QD, it can be used alone or in combination with MTX
Pfizer Korea (CEO Dong-wook Oh) ​​announced on the 10th that it has received approval for Xeljanz XR 11 mg, a rheumatoid arthritis treatment, from the MFDS on the 7th.

Xeljanz XR is a sustained-release tablet formulation of the existing Xeljanz 5mg (Tofacitinib). It can be used for the treatment of moderate to severe active rheumatoid arthritis in adults who do not respond adequately to MTX or are not tolerated.

Xeljanz, an oral JAK inhibitor, inhibits the JAK signaling pathway (Jak-STAT pathway), which is involved in the production of cytokines that cause inflammation in the body. Following the US in 2012, it was approved in Korea as a treatment for rheumatoid arthritis in 2014.

Since then, the i
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