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  • Big Pharmas busy reaching out for KRAS targeted therapy
  • by Kim, Jin-Gu | translator Byun Kyung A | Jan 18, 2021 06:14am
Considered impossible technology for 40 years, but recently showed plausible clinical findings
Amgen and Mirati leading the R&D race, Novartis, Sanofi, Merck and Bayer starts preclinical

Global pharmaceutical giants are eager to develop targeted therapy for ¡®Kirsten rat sarcoma viral oncogene homolog (KRAS)¡¯ mutation, initially considered as an impenetrable technology for last four decades.

Apparently, KRAS mutation is found in about one out of four cancer types. Specifically, the mutation is frequently found in cancer types with bad prognosis like lung cancer, colon cancer and pancreatic cancer.

Pioneered by Amgen, small and big companies like Novartis, Sanofi, Bayer, Boehringer Ingelheim, Merck and Mirati Therapeutics are fiercely competing against each other to dominate the blue ocean.

¡ßWhy did MSD bet USD 2.5 billion on candidate medicine in preclinical trial phase?

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