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  • Targeted therapies for HER2m NSCLC actively developed
  • by Son, Hyung-Min | translator Kang, Shin-Kook | Jun 18, 2024 05:49am
Various companies have started developing drugs for HER2-mutant non-small-cell lung cancer
Boehringer Ingelheim¡¯s candidate drug shows effect in trial¡¦Yuhan Corp starts clinical trial
Hanmi Pharmaceutical reattempts anticancer drug development after failing with poziotinib
The domestic and foreign pharmaceutical industry has taken up the challenge of developing a new drug for HER2-positive NSCLC. After Enhertu opened the door by obtaining the first marketing authorization as an anticancer drug targeting the HER2 mutation in Korea, many later entrants such as Yuhan Corp, Boehringer Ingelheim, and Hanmi Pharmaceutical have also started clinical trials.

Until now, there have been a number of drugs targeting various gene mutations such as EGFR, ALK, ROS1, BRAF, MET, and RET in NSCLC, but none has targeted HER2. Approximately 2-4% of patients with NSCLC have a HER2 mutation. Due to its low prevalence, the companies had difficulty developing targeted therapies.

This is why the clinical res
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